Abstract Background Left ventricular hypertrophy (LVH) is most common when driven by hypertension, and it is a strong independent risk factor for adverse cardiovascular events and death. Some animal models support a role for gut microbiota and metabolites in the development of LVH, but cohort studies confirming these findings in populations are lacking. Methods and Results We investigated the alterations of gut microbiota and metabolites in 30 patients with hypertension, 30 patients with hypertensive LVH, and 30 matched controls on the basis of 16S rDNA and metabolomic analyses. Thirty stool and 90 serum samples were collected in fasting conditions. ANOVA/Kruskal–Wallis/Pearson's χ^2/Fisher's exact test and Bonferroni's correction were used (P<0.0167) for comparison among the 3 groups. A regression analysis and subgroup analysis were performed between gut microbiota and left ventricular mass index (LVMI) and metabolites and LVMI, respectively. Spearman correlation analysis was performed between metabolites and flora and metabolites and LVMI. We observed LVH‐enriched Faecalitalea (β=6758.55 [95% CI, 2080.92–11436.18]; P=0.009), Turicibacter (β=8424.76 [95% CI, 2494.05–14355.47]; P=0.01), Ruminococcus torques group (β=840.88 [95% CI, 223.1–1458.67]; P=0.013), and Erysipelotrichaceae UCG‐003 (β=856.37 [95% CI, 182.76–1529.98]; P=0.019) were positively correlated with LVMI. A total of 1141 (in sera) and 2657 (in feces) metabolites were identified. There was a sex‐specific association between metabolites and LVMI. Significant changes in metabolic pathways in LVH were also observed, especially bile acid and lipid metabolism pathways. Conclusions Our study demonstrated the disordered gut microbiota and microbial metabolite profiles in LVH. This highlights the roles of gut bacteria and metabolite in this disease and could lead to new intervention, diagnostic, or management paradigms for LVH. Registration URL: [32]https://www.chictr.org.cn; Unique Identifier: ChiCTR2200055603. Keywords: gut microbiota, hypertension, left ventricular hypertrophy, metabolomics Subject Categories: Hypertension, Biomarkers, Metabolism, Remodeling __________________________________________________________________ Nonstandard Abbreviations and Acronyms BA bile acid CDCA chenodeoxycholic acid DA differential abundance DCA deoxycholic acid F/B Firmicutes/Bacteroidetes KEGG Kyoto Encyclopedia of Genes and Genomes LA linolenic acid LDA linear discriminant analysis LVMI left ventricular mass index PLS‐DA partial least squares discrimination analysis TMAO trimethylamine N‐oxide Clinical Perspective. What Is New? * Microbial profiles of patients with left ventricular hypertrophy in the real world, the metabolite signature profiles, and microbial biomarkers for early detection of left ventricular hypertrophy. What Are the Clinical Implications? * Our study can provide ideas for early intervention targets to prevent patients with hypertension from developing left ventricular hypertrophy and to provide possible means of reversal for patients who have already developed left ventricular hypertrophy. Hypertension is a leading risk factor for death and strongly related to cerebrovascular and cardiovascular disease.[33] ^1 , [34]^2 The pathophysiological mechanisms of essential hypertension remain largely unknown, which hinders the development of targeted therapies. Pathological left ventricular hypertrophy (LVH) is most common when driven by hypertension, and it is a strong independent risk factor for adverse cardiovascular events and death, even when left ventricular systolic function is normal and there is no preceding myocardial infarction.[35] ^3 Therefore, timely diagnosis and early treatment are the keys. It is well documented that treatment of hypertension is a means of delaying the development of LVH.[36] ^4 , [37]^5 LVH does not seem to be entirely caused by blood pressure (BP). Clinical treatment has confirmed that although some patients with hypertension have good long‐term BP control, the hypertrophic left ventricle is difficult to return to normal.[38] ^6 Animal studies have demonstrated that some spontaneously hypertensive rats develop ventricular hypertrophy before the increase of BP.[39] ^7 There is mounting evidence to suggest that the gut microbiome plays an important role in the development and pathogenesis of hypertension.[40] ^8 Therefore, we believe that hypertensive LVH is not only a simple process of cell volume increase and corresponding subcellular structural changes caused by hemodynamic overload but also a reasonable remodeling process of myocardial structure, function, and metabolism under the regulation of neurohumoral factors.[41] ^9 , [42]^10 , [43]^11 We sought to identify new intervention targets for the treatment and reversal of LVH through a novel approach to reduce the adverse outcomes of hypertensive LVH, the risk of heart failure, and the hospitalization rate of heart failure. The gut microbiota plays an important role in maintaining human health; it interacts with the host, and each influences the other.[44] ^12 Imbalances in the composition and function of these gut microbes are linked to many diseases, such as obesity,[45] ^13 diabetes,[46] ^14 metabolic syndrome,[47] ^15 cardiovascular disease,[48] ^16 and other chronic diseases. The gut microbiota mediates microbiome–host genomic cross‐talk by sending biological signals to the host, including microbial metabolites and proinflammatory molecules.[49] ^17 Metabolic remodeling is a precursor to most other pathological changes and may play an important role in cardiac hypertrophy and heart failure.[50] ^7 , [51]^18 , [52]^19 During hypertensive LVH, metabolic changes have been observed in the cardiac muscle, which prefers to convert from fatty acids to glucose to produce ATP.[53] ^7 Short‐chain fatty acids are reported to affect host physiology and the cardiovascular system and are thought to play a part in regulating blood pressure.[54] ^20 Organ et al[55] ^21 found that acetate supplementation significantly reduced systolic and diastolic BP, cardiac fibrosis, and LVH. There are limited studies indicating a direct association between gut microbe and metabolites and LVH, especially in clinical trials. There are some important gaps in knowledge about the gut and LVH that remain unexplored, and critical issues that should be addressed, such as the microbial profiles of patients with LVH in the real world, the metabolite signature profiles, and microbial biomarkers for early detection of LVH. Our study aimed to address the following issues: (1) to find alterations in microbial profiles and metabolite profiles of LVH; (2) to identify potential biomarkers for early detection of LVH populations in clinical trials; (3) to determine the relationship between gut microbe and metabolites; and (4) to identify the metabolic pathways involved in LVH and hypertension. Our study can provide ideas for early intervention targets to prevent patients with hypertension from developing LVH and to provide possible means of reversal for patients who have already developed LVH. METHODS Data Availability Statement To minimize the possibility of unintentionally sharing information that can be used to reidentify private information, a subset of the data generated for this study is available at the National Center for Biotechnology Information under the BioProject and can be accessed at [56]https://www.ncbi.nlm.nih.gov/bioproject/1065087. All untargeted metabolomic data used in this publication have been deposited to the European Molecular Biology Laboratory–European Bioinformatics Institute MetaboLights database with the identifier MTBLS9381 (fecal metabolomics) and MTBLS9370 (serum metabolomics). The complete data set can be accessed at [57]https://www.ebi.ac.uk/metabolights/MTBLS9370 and [58]https://www.ebi.ac.uk/metabolights/MTBLS9381. Participants The study was conducted in the Second Affiliated Hospital of Baotou Medical College, Inner Mongolia, China, between November 8, 2021, and July 1, 2022. Our study recruited 90 participants, including 30 patients with hypertension, 30 patients with hypertensive LVH, and 30 self‐reported healthy subjects (controls). All 3 groups were matched for sex and age. Clinical information was collected, including age, sex, height, weight, body mass index, systolic BP, diastolic (BP), heart rate, fasting blood glucose, triglycerides, total cholesterol, high‐density lipoprotein, low‐density lipoprotein, uric acid, creatinine, blood routine, history of antihypertensive medication, history of smoking, and alcohol status. Individuals were excluded if they had secondary hypertension; were hospitalized for acute myocardial infarction or unstable angina pectoris with coronary angiography stenosis >50%; had previous revascularization surgery (percutaneous coronary intervention or coronary artery bypass grafting); had acute or chronic heart failure; had valvular heart disease, dilated or hypertrophic cardiomyopathy, rheumatic heart disease, or congenital heart disease; had diabetes; had severe liver or kidney disease or dialysis; had serum creatinine >221 mol/L (>2.5 mg/dL); had a malignant tumor; had infections, diarrhea, and anti‐inflammatory use in the past week; or had other inflammatory diseases. Fecal and plasma samples were collected for comparison of gut microbial communities using 16S rDNA and of metabolites using nontargeted metabolomics (liquid chromatography–mass spectrometry). Feces and plasma samples were collected at the hospital and stored immediately at −80 °C until processing. Only 30 stool specimens were collected, 10 from each group; 90 blood samples were collected. All subjects signed informed consent forms. The present study was approved by the local ethics committee (LW‐018). This study followed the Strengthening the Reporting of Observational Studies in Epidemiology cohort reporting guidelines.[59] ^22 Measurement of Blood Pressure and Cardiac Structure Resting BP was measured by experienced physicians, and the average of 3 readings was taken as our measure of BP. Hypertension was defined as systolic BP ≥140 mm Hg or diastolic BP ≥90 mm Hg or a previous diagnosis of hypertension.[60] ^23 All participants underwent full M‐type, 2‐dimensional, and Doppler echocardiographic examinations, which were performed by the same well‐trained physician who was blind to the participants' grouping. The physician used a VIVID S70n ultrasound system and M5Sc probes, and the patient was breathing quietly in the left‐lying position. The following echocardiographic parameters were collected: left ventricular end‐diastolic diameter, left ventricular posterior wall thickness, and interventricular septal thickness. The left ventricular mass index (LVMI) was calculated as left ventricular mass divided by body surface area. LVH was defined according to the 2013 European Society of Hypertension/European Society of Cardiology guidelines for the management of arterial hypertension[61] ^24 : LVMI >95 g/m^2 in women and >115 g/m^2 in men. The formulations are as follows: graphic file with name JAH3-13-e034230-e004.jpg [MATH: Body surface area=0.007184×heightcm×0.125×weightkg×0.425m2 :MATH] [MATH: LVMI(g/m2)=left ventricularend‐diastolic diameterg/body surface area(m2) :MATH] 16S rDNA Total genome DNA from samples were extracted using a Magnetic Soil and Stool DNA Kit (Tiangen Biotech, Beijing, China). DNA concentration and purity were monitored on 1% agarose gels. According to the concentration, DNA was diluted to 1 ng/μL using sterile water. 16S rRNA genes were amplified using the specific primer with the barcode. All polymerase chain reaction (PCRs) were carried out in 30‐μL reactions with 15 μL of Phusion High‐Fidelity PCR Master Mix (New England Biolabs, Ipswich, MA); 0.2 μmol/L of forward and reverse primers, and about 10 ng template DNA. Thermal cycling consisted of initial denaturation at 98 °C for 1 minute, followed by 30 cycles of denaturation at 98 °C for 10 seconds, annealing at 50 °C for 30 seconds, and elongation at 72 °C for 30 seconds and finally 72 °C for 5 minutes. The same volume of 1X loading buffer (containing SYBR green) was mixed with PCR products and electrophoresis on 2% agarose gel operated for detection. Samples with bright main strips between 400 and 450 bp were chosen for further experiments. PCR products were mixed in equidensity ratios. Then, a mixture of PCR products was purified with Qiagen Gel Extraction Kit (Qiagen, Venlo, The Netherlands). Sequencing libraries were generated using TruSeq DNA PCR‐Free Sample Preparation Kit (Illumina, San Diego, CA) following manufacturer's recommendations and index codes were added. The library quality was assessed on the Qubit@ 2.0 Fluorometer (Thermo Scientific, Waltham, MA) and Agilent Bioanalyzer 2100 system (Agilent Technologies, Santa Clara, CA). At last, the library was sequenced on an Illumina NovaSeq6000 platform and 250‐bp paired‐end reads were generated. Paired‐end reads from the original DNA fragments were merged using FLASH, which was designed to merge paired‐end reads when at least some of the reads overlap the read generated from the opposite end of the same DNA fragment. Paired‐end reads were assigned to each sample according to the unique barcodes. Metabonomics The plasma and fecal samples were thawed at 4 °C, and 100‐μL aliquots were mixed with 400 μL of cold methanol/acetonitrile (1:1, v/v) to remove the protein. The mixture was centrifuged for 20 minutes (14 000g, 4 °C). The supernatant was dried in a vacuum centrifuge. For liquid chromatography–mass spectrometry analysis, the samples were redissolved in 100 μL acetonitrile/water (1:1, v/v) solvent and centrifuged at 14 000g at 4 °C for 15 minutes, and then the supernatant was injected. Analysis was performed using an ultra‐high‐performance liquid chromatography (Vanquish UHPLC, Thermo) coupled to a quadrupole time‐of‐flight (TripleTOF 6600; AB Sciex, Concord, ON, Canada) in Shanghai Applied Protein Technology Co., Ltd. For hydrophilic interaction liquid chromatography separation, samples were analyzed using a 2.1 mm×100 mm Acquity UPLC BEH Amide 1.7‐μm column (Waters Corp., Wexford, Ireland). In both electrospray ionization–positive and –negative modes, the mobile phase contained A=25 mmol/L ammonium acetate and 25 mmol/L ammonium hydroxide in water and B=acetonitrile. The gradient was 98% B for 1.5 minutes and was linearly reduced to 2% in 10.5 minutes, and then kept for 2 minutes, and then increased to 98% in 0.1 minute, with a 3‐minute reequilibration period employed. The electrospray ionization source conditions were set as follows: Ion Source Gas1 as 60, Ion Source Gas2 as 60, and curtain gas as 30; source temperature: 600 °C, IonSpray Voltage Floating±5500 V. In mass spectrometry–only acquisition, the instrument was set to acquire over the m/z range 80 to 1200 Da, the resolution was set at 60 000, and the accumulation time was set at 100 milliseconds. In auto tandem mass spectrometry acquisition, the instrument was set to acquire over the m/z range 70 to 1200 Da, the resolution was set at 30 000, and the accumulation time was set at 50 milliseconds and excluded time within 4 seconds. The raw mass spectrometry data were converted to MzXML files using ProteoWizard MSConvert before importing into freely available XCMS software. For peak picking, the following parameters were used: centWave m/z=10 ppm, peakwidth=c (10, 60), prefilter=c (10, 100). For peak grouping, bw=5, mzwid=0.025, minfrac=0.5 were used. CAMERA (Collection of Algorithms of MEtabolite pRofile Annotation) was used for annotation of isotopes and adducts. In the extracted ion features, only the variables having >50% of the nonzero measurement values in at least 1 group were kept, and then the nonzero measurement values were filled by knn algorithm. Compound identification of metabolites was performed by comparing of accuracy m/z value (<10 ppm) and tandem mass spectrometry spectra with an in‐house database established with available authentic standards. Statistical Analysis Statistical analyses were performed using R software (R Foundation for Statistical Computing, Vienna, Austria). Normally distributed variables were expressed as mean±SD, and the ANOVA test was used; abnormally distributed variables were shown as the median (quartile), and nonparametric (Kruskal–Wallis) tests were used. Categorical data were expressed as the numbers and percentages, using Pearson's χ^2 test or Fisher's exact test, as appropriate. Multiple testing correction was performed using Bonferroni correction, and the significance of the P value was assessed at 0.0167 (0.05/3), as pairwise comparisons were performed 3 times among the 3 groups. A multivariable linear regression analysis was performed between specific gut microbiota and LVMI. Multivariate‐adjusted models were used: model 1: adjusted age and sex; model 2=model 1+body mass index+low‐density lipoprotein+total cholesterol+fasting blood glucose+history of antihypertensive medication. Spearman correlation analysis was performed to determine the correlation between differential metabolites and differential flora and the correlation between metabolites and LVMI. Subgroup analyses were also used to investigate the sex differences in associations between metabolites and LVMI. Sequences analyses were performed with UPARSE software package using the UPARSE‐OTU and UPARSE‐OTUref algorithms. In‐house Perl scripts were used to analyze α (within samples) and β (among samples) diversity. Sequences with ≥97% similarity were assigned to the same operational taxonomic units (OTUs). We pick a representative sequence for each OTU and use the RDP classifier to annotate taxonomic information for each representative sequence (Silva 132; [62]https://www.arb‐silva.de/). Rarefaction curves were generated on the basis of these 3 metrics. Graphical representation of the relative abundance of bacterial diversity from phylum to species can be visualized using Krona chart. Principal component analysis was applied to reduce the dimension of the original variables using the QIIME software package. QIIME calculates both weighted and unweighted unifrac distance, which are phylogenetic measures of β diversity. We used weighted unifrac distance for principal coordinate analysis. Linear discriminant analysis (LDA) effective size was used for the quantitative analysis of biomarkers within different groups. LDA effective size >2 and P value <0.05 were used to screen significantly changed bacteria. Analysis of similarities and permutational multivariate ANOVA were performed on the basis of the Bray–Curtis dissimilarity distance matrices to identify differences of microbial communities between the 2 groups. After sum normalization, the processed metabolomics data were analyzed by the R package ropls, where it was subjected to multivariate data analysis, including Pareto‐scaled principal component analysis, partial least‐squares discrimination analysis (PLS‐DA), and orthogonal PLS‐DA. The 7‐fold cross‐validation and response permutation testing were used to evaluate the robustness of the model. The variable importance in the projection value of each variable in the orthogonal PLS‐DA model was calculated to indicate its contribution to the classification. The Kruskal–Wallis test with post hoc multiple comparison was applied to determine the significance of differences among 3 groups of independent samples. Variable importance in the projection >1 and P value <0.05 were used to screen significantly changed metabolites. All identified metabolites were mapped to the Kyoto Encyclopedia of Genes and Genomes (KEGG) database to find general biochemical pathways ([63]http://geneontology.org/). The KEGG pathway enrichment analysis was performed using MBROLE version 2.0 ([64]http://csbg.cnb.csic.es/mbrole2/). KEGG differential abundance (DA) score plots were performed by ggplot2 package (R software). DA score is calculated by first applying a nonparametric DA test to all metabolites in a pathway. Then, after determining which metabolites are significantly increased/decreased in abundance, the DA score is defined as[65] ^25 : [MATH: No.of metabolites increasedNo.of metabolites decreasedNo.of measured metabolites in pathway :MATH] A score of 1 indicates all measured metabolites in the pathway increase, and − 1 indicates all measured metabolites in a pathway decrease. RESULTS Clinical Features of the Cohort Our cohort recruited 30 patients with hypertension, 30 patients with LVH, and 30 self‐reported healthy subjects, aged 63.9±8.3 years, 37 of whom were women (41.1%). The clinical characteristics of the cohort are shown in Table [66]1. We must acknowledge that power is low with so few people. No differences were observed among groups concerning the age, sex, height, body mass index, total cholesterol, triglycerides, high‐density lipoprotein, low‐density lipoprotein, fasting blood glucose (FBG), heart rate, and alcohol status. systolic BP, diastolic BP, smoking status, left ventricular end‐diastolic diameter, interventricular septal thickness, left ventricular posterior wall thickness, left ventricular end‐diastolic diameter and LVMI were significantly different among the 3 groups. Table 1. Demographics and Clinical Features of the Cohort Variables Total (n=90) LVH (n=30) Hypertension (n=30) Control (n=30) P value Sex, n (%) 0.725 Male 53 (58.9) 18 (60) 19 (63.3) 16 (53.3) Female 37 (41.1) 12 (40) 11 (36.7) 14 (46.7) Age, y 63.9±8.3 64.1±9.1 64.0±8.0 63.5±8.0 0.963 Smoking, n (%) 0.001 No 65 (72.2) 17 (56.7) 19 (63.3) 29 (96.7) Yes 25 (27.8) 13 (43.3) 11 (36.7) 1 (3.3) Alcohol status, n (%) 0.067 No 72 (80.0) 21 (70) 23 (76.7) 28 (93.3) Yes 18 (20.0) 9 (30) 7 (23.3) 2 (6.7) History of hypertension medication, n (%) <0.001 No 31 (34.4) 1 (3.3) 0 (0) 30 (100) Yes 59 (65.6) 29 (96.7) 30 (100) 0 (0) Height, cm 166.4±7.2 168.0±7.5 166.6±7.2 164.6±6.6 0.195 Weight, kg 68.8±12.1 72.4±13.7 69.6±12.1 64.5±9.2 0.037 Body mass index, kg/m^2 24.7±3.2 25.6±3.9 24.9±3.1 23.7±2.4 0.076 Total cholesterol, mmol/L 4.6±0.9 4.7±0.9 4.4±1.0 4.8±0.7 0.175 Triglycerides, mmol/L 1.4 (1.0–1.9) 1.7 (1.1–2.1) 1.4 (1.1–1.9) 1.1 (0.8–1.6) 0.125 HDL, mmol/L 1.3 (1.0–1.6) 1.1 (1.0–1.5) 1.2 (1.0–1.5) 1.4 (1.2–1.8) 0.061 LDL, mmol/L 2.9±0.8 3.0±0.8 2.8±0.9 2.9±0.6 0.589 Fasting blood glucose, mmol/L 5.4±0.7 5.3±0.7 5.2±0.6 5.7±0.8 0.016 Creatinine, mmol/L 73.6±17.1 75.9±20.5 75.3±12.6 69.3±17.5 0.285 Uric acid, mmol/L 317.0±85.5 282.7±73.4 319.3±77.3 322.1±97.0 0.589 Systolic BP, mm Hg 135.0 (125.0–143.8) 141.5 (136.0–150.0) 140.0 (127.0–144.0) 122.5 (114.0–130.8) <0.001 Diastolic BP, mm Hg 82.8±12.6 88.6±11.6 85.0±13.4 74.7±8.1 <0.001 Heart rate, beats 76.4±10.3 78.3±10.3 74.8±10.2 76.2±10.5 0.409 LVDD, mm 4.7 (4.4–4.9) 4.8 (4.6–5.3) 4.6 (4.3–4.8) 4.5 (4.3–4.8) <0.001 Interventricular septal thickness, mm 1.0 (0.9–1.1) 1.2 (1.1–1.4) 0.9 (0.8–1.0) 0.9 (0.8–0.9) <0.001 LVPWT, mm 0.9 (0.8–1.0) 1.0 (1.0–1.2) 0.9 (0.8–1.0) 0.8 (0.8–0.9) <0.001 LVM, g 146.7 (123.1–181.8) 219.4 (177.5–254.6) 137.7 (123.0–151.4) 125.5 (113.6–142.5) <0.001 0.008 LVMI, g/m^2 91.8±25.3 121.4±18.8 78.7±10.8 75.3±11.3 <0.001 [67]Open in a new tab Data are presented as mean±SD, n (%), or median (quartile). Normally distributed variables were used for ANOVA test, abnormally distributed variables were used for nonparametric tests (Kruskal–Wallis test); χ^2 or Fisher test for categorical variables. Normality was examined using the Shapiro–Wilk test. Bonferroni's correction was applied (0.05/3=0.0167). BP indicates blood pressure; HDL, high‐density lipoprotein; LDL, low‐density lipoprotein; LVDD, left ventricular end‐diastolic diameter; LVH, left ventricular hypertrophy; LVM, left ventricular mass; LVMI, left ventricular mass index; and LVPWT, left ventricular posterior wall thickness. Gut Microbial Rarefaction of samples to 55 000 reads showed consistent and plateauing diversity metrics across samples (Figure [68]S1). The top 10 differentially enriched bacterial taxa of each group are presented in our study. At the phylum level, hypertension, LVH, and control group, all presented Firmicutes and Bacteroidetes as the major. Compared with the control group, the proportion of Firmicutes and Actinobacteria increased the most in the LVH group, followed by the hypertension group. However, Bacteroidetes was significantly reduced in the LVH group, followed by the hypertension group. In addition, Proteobacteria and Tenericutes were significantly decreased in the LVH group and significantly increased in the hypertension group, while Verrucomicrobia was significantly increased in the LVH group and significantly decreased in the hypertension group. An increased ratio of Firmicutes/Bacteroidetes (F/B) in the gut microbiota of both individuals with LVH and individuals with hypertensive compared with controls was found, resulting from a reduction of Bacteroidetes and an enrichment of Firmicutes (Figure [69]1). More detailed taxonomic levels are shown in Figures [70]S2 through [71]S7. The above results indicate that the imbalanced structure of the intestinal flora in patients with LVH and hypertension and the alterations of some intestinal flora of the 2 groups were different, suggesting that these changes of gut microbiata increase the susceptibility to LVH. Figure 1. The top 10 differentially enriched bacterial taxa of each group at phylum level. Figure 1 [72]Open in a new tab HP indicates hypertension; and LVH, left ventricular hypertrophy. The microbial β diversity (between samples) and α diversity (within samples) metrics were quantified in our study. We observed an elevation in bacterial Chao and Abundance‐Based Coverage Estimator richness in the LVH group, although the difference was not statistically significant (P>0.05; Table [73]S1, Figure [74]S8), which may suggest the overgrowth of a variety of harmful bacteria in patients with LVH. There was no association between α diversity and LVMI and BP (data not shown). The microbial β diversity showed no significant differences in gut microbiome composition among the 3 groups (Figure [75]2, Figure [76]S9). Some specific taxa in control, hypertension, or LVH groups were prevalent, detailed by LDA effective size (Figure [77]3A through [78]3C). We detected a total of 44, 16, and 13 biomarkers with LDA scores >2 that were significantly different between the LVH group and controls, the hypertension group and controls, and the LVH and hypertension groups, respectively. Of these, the specific taxa with the highest LDA score in LVH belongs to Firmicutes, and in controls and hypertension belong to Bacteroidetes. At the genus level, we identified that individuals with LVH had higher levels of genera such as Streptococcus, Romboutsia, Lactobacillus, Rothia, Granulicella, Marmoricola, Enorma, Leuconostoc, Peptoniphilus, Faecalitalea, Turicibacter, Desulfovibrio, Uruburuella, Ruminococcus torques group, and Erysipelotrichaceae UCG‐003, while subjects with hypertension had higher levels of Lactobacillus, Granulicatella, and Eubacterium coprostanoligenes group, healthy participants had higher levels of Roseburia, Acetitomaculum, Fournierella, Odoribacter, Prevotella 2, Christensenellaceae R7 group, Eubacterium ruminantium group, GCA_900 066 575, Lachnospira, Lachnospiraceae NK4A136 group, and Lachnospiraceae UCG‐010. Figure 2. Comparison of the microbial β diversity (as accessed by principal coordinate analysis used weighted unifrac distance) in the 3 groups. Figure 2 [79]Open in a new tab ANOSIM (analysis of similarities) is a nonparametric test based on the Bray–Curtis algorithm. R>0 indicates significant differences between groups, R<0 indicates significant difference within the group is greater than the difference between the groups. ADONIS is known as permutational multivariate ANOVA or nonparametric multivariate ANOVA. The F score ranges from 0 to 1, with the higher the value, the better the model performance. Top left: LVH vs HP vs control; bottom left: LVH vs HP; top right: LVH vs control; bottom right: HP vs control. HP indicates hypertension; and LVH, left ventricular hypertrophy. Figure 3. Linear discriminant analysis effect size (LEfSe) of each cohort to visualize differences in bacterial species. Figure 3 [80]Open in a new tab A, LVH vs control; B, LVH vs HP; and C, HP vs control. LEfSe LDA>2 and P value<0.05 were used to screen significant changed bacteria. HP indicates hypertension; and LVH, left ventricular hypertrophy. We performed correlations between the microbiome and LVMI (Table [81]2, Table [82]S2). LVH‐enriched Faecalitalea (β=6758.55 [95% CI, 2080.92–11436.18]; P=0.009), Turicibacter (β=8424.76 [95% CI, 2494.05–14355.47]; P=0.01), Ruminococcus torques group (β=840.88 [95% CI, 223.1–1458.67]; P=0.013), and Erysipelotrichaceae UCG‐003 (β=856.37 [95% CI, 182.76–1529.98]; P=0.019) were positively correlated with LVMI, but control‐enriched GCA.900066575 (β=−46478.71 [95% CI=−90661.93 to −2295.49]; P=0.049) was negatively linked to LVMI. After adjusting for 2 models, only Faecalitalea (β=6077.34 [95% CI, 1633.86–10520.82]; P=0.014), Ruminococcus torques group (β=853.73 [95%CI, 283.14–1424.32]; P=0.008), and Erysipelotrichaceae UCG‐003 (β=880.05 [95% CI, 282.6–1477.5]; P=0.009) remained statistically significantly associated with LVMI. It is worth noting that the bacteria genera that distinguish LVH from the hypertension group were Faecalitalea, Erysipelotrichaceae UCG‐003, Ruminococcus torques group, and Turicibacter, which were highly expressed in LVH. Table 2. Relationship Between Gut Microbiota and LVMI Model 1, β (95% CI); P value Model 2, β (95% CI); P value Turicibacter 8424.76 (2494.05 to 14355.47); 0.01 5770.46 (−1347.22 to 12888.13); 0.127 Faecalitalea 6758.55 (2080.92 to 11436.18); 0.009 6077.34 (1633.86 to 10520.82); 0.014 Enorma 124337.08 (4889.52 to 243784.63); 0.052 94315.07 (−26841.66 to 215471.8); 0.142 Ruminococcus torques group 840.88 (223.1 to 1458.67); 0.013 853.73 (283.14 to 1424.32); 0.008 Erysipelotrichaceae UCG‐003 856.37 (182.76 to 1529.98); 0.019 880.05 (282.6 to 1477.5); 0.009 GCA.900066575 −46478.71 (−90661.93 to −2295.49); 0.049 −31365.99 (−80514.88 to –17782.9); 0.225 [83]Open in a new tab Model 1: adjusted for age and sex; model 2=Model 1+body mass index; low‐density lipoprotein; total cholesterol; fasting blood glucose; history of antihypertensive medication. LVMI indicates left ventricular mass index. Metabolomics (Feces and Plasma) Many metabolites of the gut microbiota serve as microbe–host bridges and can influence host physiology either in the gut or through entry into the bloodstream. Therefore, the levels of the intestinal metabolic profiling from feces and plasma were both measured in our study. A subset of 30 participants (10 from each group) from the present study were enrolled in the feces study (Tables [84]S3). PLS‐DA and orthogonal PLS‐DA under both positive ion (ES+) and negative ion (ES−) modes succeed in distinguishing samples of plasma and fecal metabolomics between the LVH and control groups, the LVH and hypertension groups, and the hypertension and control groups (Figures [85]4A and [86]4B; Figures [87]5A and [88]5B). Variable importance in the projection plots were also provided (Figures [89]S10 and [90]S11). The metabolites of 3 groups were identified in ES+ and ES− mode, and the metabolites of the 3 groups were significantly different (Figure [91]6). These results indicated that LVH and hypertension significantly altered the intestinal flora metabolic profiles. Figure 4. PLS‐DA score plots based on the metabolic profiles from the control, LVH, and HP groups in ES+ and ES−. Figure 4 [92]Open in a new tab A, In plasma samples; and B, in feces samples. The 7‐fold cross‐validation and response permutation testing were used to evaluate the robustness of the model. ES+ indicates positive ion; ES–, negative ion; HP, hypertension; LVH, left ventricular hypertrophy; and PLS‐DA, partial least‐squares discriminant analysis. Figure 5. OPLS‐DA score plots based on the metabolic profiles from the control, LVH, and HP groups in ES+ and ES−. Figure 5 [93]Open in a new tab A, In plasma samples; and (B) in feces samples. The 7‐fold cross‐validation and response permutation testing were used to evaluate the robustness of the model. ES+ indicates positive ion; ES–, negative ion; HP, hypertension; LVH, left ventricular hypertrophy; and OPLS‐DA, orthogonal partial least‐squares discriminant analysis. Figure 6. Venn diagram shows the number of altered metabolites in plasma and feces samples from the control, LVH, and HP groups in ES+ and ES−. Figure 6 [94]Open in a new tab ES+ indicates positive ion; ES–, negative ion; HP, hypertension; and LVH, left ventricular hypertrophy. In plasma tests, a total of 1141 metabolites were identified. A total of 132 (ES+ mode, 72; ES− mode, 60) and 49 (ES+ mode, 20; ES− mode, 29) metabolites were significantly different between the LVH and control groups and the LVH and hypertension groups, respectively. In addition, 116 (ES+ mode, 66; ES− mode, 50) serum metabolites were significantly different between hypertension and controls. Of these, the majority were lipids and lipid‐like molecules. The expression of the lipids and lipid‐like molecules was downregulated in both LVH and hypertension. Inversely, the majority of the organic acids and derivatives and organoheterocyclic compounds were upregulated in LVH and hypertension (Figures [95]7A and [96]7C, Tables [97]S4 and [98]S5). Notably, metabolites such as bile acids (BAs), trimethylamine N‐oxide (TMAO), linolenic acid (LA), and choline were significantly changed in patients with LVH. The free BAs of deoxycholic acid (DCA) was significantly upregulated, while the contents of conjuncted BAs such as glycocholic acid was significantly downregulated. In addition, the content of TMAO and choline in LVH was significantly upregulated, while LA in LVH was significantly downregulated. TMAO is derived mainly from the oxidation of trimethylamine by the gut flora. Intestinal microorganisms metabolize the ingested lecithin and choline and produce trimethylamine, which is then oxidized by flavin monooxygenase 3 or other flavin monooxygenase to produce TMAO.[99] ^26 Both BAs and TMAO have been found to be involved in the occurrence and development of hypertension, cardiovascular disease, diabetes, and other diseases, and may be related to inflammatory response.[100] ^27 , [101]^28 , [102]^29 , [103]^30 , [104]^31 , [105]^32 Inflammation and oxidative stress are the main factors causing BP increase and organ damage, such as LVH, in hypertension. This is a possible reason for the changes in BAs and TMAO levels in patients with LVH. LA and α‐LA, are essential fatty acids that have been shown to have a variety of beneficial effects, including antimetabolic syndrome effects, antimetabolic syndrome, anticancer, antiinflammatory, antioxidant, antiobesity, neuroprotection, and regulation of the intestinal flora properties.[106] ^33 Figure 7. The relative amount of plasma metabolites varied in the LVH, HP, and control groups. Figure 7 [107]Open in a new tab A, LVH vs HP; B, LVH vs control; and C, HP vs control. Variable importance in the projection >1 and P value <0.05 were used to screen significant changed metabolites. HP indicates hypertension; and LVH, left ventricular hypertrophy. In fecal metabolite tests, a total of 2657 metabolites were identified. Seventy‐four (ES+ mode, 53; ES− mode, 21) and 59 (ES+ mode, 31; ES− mode, 28) fecal metabolites were significantly different between LVH and controls and LVH and hypertension, respectively. Additionally, 95 (ES+ mode, 69; ES− mode, 26) fecal metabolites were significantly different between the hypertension and controls. Different from the differential metabolites in blood, organic acids and derivatives were mostly found in feces. The expression of the lipids and lipid‐like molecules were downregulated in the LVH group compared with the hypertension group, but its expression was upregulated in the LVH group compared with the controls. Lipids and lipid‐like molecules were down‐expressed in the LVH group compared with the controls and up‐expressed when compared with the hypertension group. When compared with controls, organic acids and derivatives were upregulated and organoheterocyclic compounds were downregulated in the hypertension group (Figure [108]8A through [109]8C; Tables [110]S6 and [111]S7). The free BAs, including DCA, chenodeoxycholic acid (CDCA), ursodeoxycholic acid, lithocholic acid, and hyodeoxycholic acid, as well as l‐homocitrulline, were significantly upregulated in patients with LVH. Homocitrulline is produced by carbamylation. Carbamylated proteins are associated with atherosclerosis.[112] ^34 A recent study found that l‐homocitrulline was associated with nonalcoholic fatty liver disease.[113] ^35 Nicotinuric acid, the main catabolite of niacin, was considered a good indicator to evaluate the biotransformation of niacin in the liver.[114] ^36 A study proved that urinary nicotinuric acid level is positively correlated with metabolic syndrome.[115] ^37 Figure 8. The relative amount of fecal metabolites varied in the LVH, HP, and control groups. Figure 8 [116]Open in a new tab A, LVH vs HP; B, LVH vs control; and C, HP vs control. Variable importance in the projection >1 and P value <0.05 were used to screen significant changed metabolites. HP indicates hypertension; and LVH, left ventricular hypertrophy. It is worth mentioning that there were metabolites identified in both serum and feces. We found 2 (zerumbone and DCA) and 1 (pregnenolone sulfate) common metabolites (with KEGG ID) both in plasma and feces between the LVH control groups and the hypertension and control groups, respectively. No common metabolites in plasma and feces were found in the LVH and hypertension groups (Figure [117]9; Tables [118]S8 through [119]S10). Zerumbone and DCA showed the same tendency both in serum and feces. However, pregnenolone sulfate showed an increased tendency in feces but decreased in serum (Figures [120]7B and [121]7C; Figures [122]8B and [123]8C). This pathogenic substance might originate from a pathway other than gut microbes.[124] ^38 Figure 9. Venn diagram of the altered metabolites shared between plasma (blue) and feces (red). Figure 9 [125]Open in a new tab A, common metabolites (with KEGG ID) both in plasma and feces between LVH and the control group; and B, common metabolites (with KEGG ID) both in plasma and feces between HP and control group. HP indicates hypertension; KEGG, Kyoto Encyclopedia of Genes and Genomes; and LVH, left ventricular hypertrophy. We examined the relationship between differential metabolites in the LVH group and LVMI and found that 131 (ES+ mode, 74; ES− mode, 57) metabolites in plasma and 56 (ES+ mode, 46; ES− mode, 10) metabolites in feces were associated with LVMI. The correlation between metabolites and LVMI differed across the sex stratification (Figures [126]S12 through [127]S15). This suggests that there was a sex‐specific association between metabolites and LVMI. Spearman correlation analysis showed that glycocholic acid and LA was significantly negatively correlated with LVMI, while hyodeoxycholic acid, CDCA, lithocholic acid, DCA, TMAO, choline, l‐homocitrulline, and nicotinuric acid were significantly positively correlated with LVMI. These metabolic variations might aggravate or even promote the pathological processes of LVH. Functional Alteration in Metabolic Pathways of Hypertension and LVH We performed an analysis based on the KEGG pathway using metabolites of DA between the LVH and control and hypertension groups to identify the metabolic pathways associated with the pathogenesis of LVH. Differential abundance scores were calculated, which captured the tendency for metabolites in a pathway to be increased/decreased relative to the control and hypertension groups. In plasma tests, compared with the control group, there were 6 and 11 significantly different metabolic pathways in the LVH and hypertension groups, respectively. Among them, 3 pathways were overrepresented in the LVH group, mainly involved in amino acid metabolism (arginine and proline metabolism), central carbon metabolism in cancer, and digestive system (protein digestion and absorption pathways); and 6 pathways were overrepresented in the hypertension group, amino acid metabolism (arginine and proline metabolism; glycine, serine, and threonine metabolism), digestive system (protein digestion and absorption, mineral absorption), central carbon metabolism in cancer, and choline metabolism in cancer (Figure [128]10). Upregulation of amino acid metabolic and protein digestion and absorption pathways has also been reported in diabetes[129] ^39 and gastric adenocarcinoma,[130] ^40 respectively. Figure 10. Functional alteration in metabolic pathways of HP and LVH. Figure 10 [131]Open in a new tab The DA score captures the average, gross changes for all metabolites in a pathway. The length of the line segment represents the absolute value of DA score, and the size of the dot at the end of the line segment represents the number of metabolites in the pathway. The larger the dot, the greater the number of metabolites. The darker the red of the line segment and the dot, the more upregulated the overall expression of the pathway, and the darker the blue, the more downregulated the overall expression of the pathway. A score of 1 indicates all measured metabolites in the pathway increase, and −1 indicates all measured metabolites in a pathway decrease. DA indicates differential abundance; HP, hypertension, and LVH left ventricular hypertrophy. It should be noted that the metabolic pathways with significant differences between LVH and hypertension in plasma tests included lipid metabolism (LA metabolism, α‐LA metabolism, biosynthesis of unsaturated fatty acids) and nervous system pathways (retrograde endocannabinoid signaling), which were significantly downregulated in the LVH group (Figure [132]9). Downregulation of the linoleic acid metabolic pathway has been reported to be associated with metabolic syndrome.[133] ^41 In addition, there were 4 significantly different metabolic pathways in fecal tests in the LVH group compared with the hypertension group, of which 2 pathways (alanine, aspartate, and glutamate metabolism; β‐alanine metabolism) were downregulated, and 1 pathway was upregulated (bile secretion) (Figure [134]10). No significantly different pathways were found in any of the other group comparisons in fecal tests (LVH versus controls, hypertension versus controls). Consistently, BA synthesis and excretion is the main pathway of cholesterol and lipid metabolism and is associated with a variety of metabolic diseases, including obesity, diabetes, and nonalcoholic fatty liver disease.[135] ^42 Correlations Between Gut Microbiome and Metabolites The significantly different metabolites in the 3 groups may be biomarkers for the development of LVH and might be derived from intestinal flora or their fermented products. To explore the association between aberrant metabolites and disordered gut microflora, we carried out a correlation analysis between differential flora and differential metabolites in plasma or feces (Figures [136]11, [137]12, [138]13, [139]14). Interestingly, we found a significant positive correlation between free BAs including DCA, hyodeoxycholic acid, CDCA, and lithocholic acid and flora including Desulfovibrio, Streptococcus, Leuconostoc, Marmoricola, and Faecalitalea, which were enriched in LVH. However, there was a significant negative correlation between these free BAs and control‐enriched Lachnospira and Lachnospiraceae NK4A136 group. On the contrary, glycocholic acid was negatively correlated with LVH‐enriched Enorma and positively correlated with control‐enriched Lachnospira and Lachnospiraceae NK4A136 group. Similarly, metabolites such as nicotinuric acid, choline, and urobilin were positively correlated with the bacteria enriched in the LVH group but negatively correlated with the bacteria in the control group. Figure 11. Correlations between metabolites in plasma and gut microbiome from the LVH and control groups. Figure 11 [140]Open in a new tab Spearman correlation analysis was used. LVH indicates left ventricular hypertrophy. Figure 12. Correlations between metabolites in feces and gut microbiome from the LVH and control groups. Figure 12 [141]Open in a new tab Spearman correlation analysis was used. LVH indicates left ventricular hypertrophy. Figure 13. Correlations between metabolites in plasma and gut microbiome from the LVH and HP groups. Figure 13 [142]Open in a new tab Spearman correlation analysis was used. HP indicates hypertension; and LVH, left ventricular hypertrophy. Figure 14. Correlations between metabolites in feces and gut microbiome from the LVH and HP groups. Figure 14 [143]Open in a new tab Spearman correlation analysis was used. HP indicates hypertension; and LVH, left ventricular hypertrophy. We examined the relationship between metabolites existing in both serum and feces, including zerumbone, DCA, and pregnenolone sulfate and microbiome. DCA in plasma and feces is positively correlated with Marmoricola, Faecalitalea, and Desulfovibrio, and inversely correlated with Lachnospira. Zerumbone in feces is positively correlated with Lachnospiraceae UCG‐010 but inversely related to Faecalitalea, Desulfovibrio, and Uruburuella. Pregnenolone sulfate in plasma was positively correlated with Odoribacter but inversely related to Eubacterium coprostanoligenes group. Pregnenolone sulfate in feces was inversely related to Fournierella (Figures [144]11 and [145]12). The close relationship between microbes and metabolites suggests that specific metabolites may be produced directly or indirectly by the corresponding gut microbes[146] ^38 and that metabolites and gut microbes may also be upstream or downstream of specific pathways, which are currently under exploration and require further validation in the future. DISCUSSION Our study revealed a novel mechanism of LVH development by intestinal flora and metabolomics. The intestinal flora composition and metabolism were significantly altered in LVH when compared with the hypertension and control groups. LVH and control participants, as well as LVH and hypertension participants, could be accurately distinguished by specific bacteria and metabolites. We found a relationship between gut microbiota and LVMI. There was a sex‐specific correlation between metabolites and LVMI. In addition, we also observed different correlations between metabolites and the flora in different groups. Furthermore, BA and lipid metabolism pathways were significantly changed during LVH development. We observed an increase in the abundance of Chao and Abundance‐Based Coverage Estimator in the LVH group, although the difference did not reach statistical significance, which may indicate the tendency of multiple harmful bacteria overgrowth in patients with LVH. β diversity of gut microbiota in the 3 groups did not exhibit any significant differences, which may suggest that the diversity and structure of gut microbiota have limited impact on the occurrence and development of LVH. It is not the composition of the whole gut microbiota but may be certain taxa that change and have effects on LVH. We found differential microbial taxa by LDA effective size analysis in the 3 groups. The second possible reason is that our sample size is not large enough to lead to insufficient statistical power. The third possible reason is that diet and the use of antihypertensive drugs changed the composition of the gut microbiome, resulting in no significant difference among the 3 groups. The shift of dominant bacteria in the gut microbiota further characterized the imbalance of LVH‐specific gut microbial environment. In the present study, bacteria such as Firmicutes and Actinobacteria increased in both the LVH and hypertension groups, while Bacteroidetes decreased. Contrary to our findings, Tsai et al[147] ^43 found that low levels of the phylum Firmicutes were associated with an increased risk of LVH. The possible reason is that their study population was diabetic, unlike our study population, which excluded people with diabetes. As shown by our study, an increased F/B ratio is represented in LVH. The specific taxa with the highest LDA score in LVH belongs to the Firmicutes phylum, and in controls and hypertension belong to the Bacteroidetes phylum. For example, at the genus level, the lactate‐producing bacteria Streptococcus and Turicibacter, both of which belong to the Firmicutes phylum, were in higher quantities in the LVH. On the contrary, acetate‐producing bacteria Prevotella, which belong to the Bacteroidetes phylum, was found to be highly accumulated in the control group. These changes in these genera may be the major contributors to the increased F/B ratio in the LVH. A higher ratio of F/B ratio has been widely considered a signature of gut dysbiosis and has been related to diabetes, hypertension, and cardiovascular disease.[148] ^44 , [149]^45 In our study, gut microbiota such as Streptococcus, Romboutsia, Lactobacillus, Rothia, Granulicella, Marmoricola, Enorma, Leuconostoc, Peptoniphilus, Faecalitalea, Turicibacter, Desulfovibrio, Uruburuella, Ruminococcus torques group and Erysipelotrichaceae UCG‐003 were typically enriched in the patients with LVH. In contrast, healthy participants had higher levels of Acetitomaculum, Fournierella, Odoribacter, Roseburia, Prevotella_2, Christensenellaceae R‐7 group, Eubacterium ruminantium group, GCA_900 066 575, Lachnospira, Lachnospiraceae NK4A136 group, and Lachnospiraceae UCG‐010. Streptococcus, a genus of gram‐positive pathological bacteria, has been shown to be associated with meningitis, pneumonia, endocarditis,[150] ^46 bowel disease,[151] ^47 cirrhosis,[152] ^48 type 1 diabetes,[153] ^49 and hypertension.[154] ^50 Roseburia is one of the major short‐chain fatty acids producer in human colon. Short‐chain fatty acids play a role in maintaining the intestinal epithelial barrier, reducing intestinal permeability, circulating lipopolysaccharide, and systemic inflammation.[155] ^51 A recent study found that several strains of Turicibacter bacteria from the mammalian gut microbiota modulate host bile and lipid compositions.[156] ^52 Some studies have found that an increased abundance of Turicibacter is associated with a high‐fat diet,[157] ^53 , [158]^54 but other studies have shown opposite relationships.[159] ^55 , [160]^56 The first reason may be that the phenotype of the Turicibacter strain is different, and the host may experience different lipid outcomes depending on its own specific Turicibacter strain. Another reason may be due to host genetic and sex changes that lead to differences in lipid responses between hosts. A third possible reason is that the effectiveness of Turicibacterium colonization is influenced by the biogeographic organization of individual microbiota.[161] ^52 An improved Streptococcus abundance was also found in simple fat people and type 1 diabetes.[162] ^49 , [163]^57 It is worth noting that certain gut microbiota play paradoxical roles like Lactobacillus. Lactobacillus, in our study, was overrepresented in both the LVH and hypertension groups. A study from a Brazilian cohort, consistent with our results, showed that in patients with hypertension, the abundance of Lactobacillus increased.[164] ^58 In addition, an increase in Lactobacillus was also observed in ST‐segment–elevation myocardial infarction.[165] ^59 However, some other studies reported the beneficial role of Lactobacillus consumption in BP regulation.[166] ^60 , [167]^61 , [168]^62 , [169]^63 The genera of Enorma, Faecalitalea, Turicibacter, Ruminococcus torques group, and Erysipelotrichaceae UCG‐003 were positively correlated with LVMI in our study. Two models were adjusted when we examined the association between microbiota and LVMI using linear models. Considering that antihypertensive drugs, lipid profile, fasting blood glucose, and body mass index may have an effect on the gut microbiome, we included them as covariates in the adjustment model. An association between Enorma and other diseases was also reported previously, such as atrial fibrillation,[170] ^64 hypertension,[171] ^61 and spinal muscular atrophy.[172] ^65 Erysipelotrichaceae UCG‐003 have been reported to be associated with inflammatory bowel diseases.[173] ^66 Metabolic profiles of both plasma and fecal samples analyzed from patients with LVH demonstrated significant alterations, which could be derived from altered bacterial functions in patients with LVH. Most importantly, our study uncovered that the expression of differential metabolite pathways are different across groups. In particular, the pathway related to BA metabolism was highly expressed in the LVH group compared with the hypertension group. This was accompanied by changes in the plasma and fecal metabolites of BAs, and BAs were significantly correlated with LVMI. Metabolites from plasma and feces, such as BAs, can act as a signaling molecule involved in glycolipid metabolism by activating the nuclear receptor farnesoid X receptor. BAs plays a role in myocardial hypertrophy, cardiomyocyte apoptosis and cardiac hemodynamic abnormalities.[174] ^67 In the present study, conjuncted BAs such as glycocholic acid were down‐expressed and free BAs including DCA, hyodeoxycholic acid, CDCA, ursodeoxycholic acid, and lithocholic acid were up‐expressed in patients with LVH. A study using Langendorff‐perfused isolated heart demonstrated the role of BAs on the heart, and the results showed that CDCA and DCA could exert positive inotropic effects by increasing cytoplasmic Ca^2+ levels in cardiomyocytes and negative isotropic effects by inhibiting sinus node activity in rat hearts within specific concentration ranges.[175] ^68 TMAO is an important metabolite of intestinal flora, which is associated with the incidence of hypertension, diabetes, obesity, and atherosclerosis.[176] ^28 The present study showed that choline and TMAO were overexpressed in LVH. It is widely known that Firmicutes and Proteobacteria are producers of trimethylamine and TMAO.[177] ^69 , [178]^70 In addition, trimethylamine and TMAO levels were associated with an increased F/B ratio.[179] ^71 , [180]^72 This provides new ideas for alleviating disease progression by downregulating the choline–trimethylamine –TMAO production pathway in gut microbiota. A meta‐analysis showed that high levels of TMAO were associated with major adverse cardiovascular events compared with low levels (risk ratio [RR] =1.62).[181] ^29 There is a dose‐dependent relationship between TMAO and the risk of death from cardiovascular disease. An animal study found cardiac remodeling in rats after TMAO intervention, with increases in left ventricular posterior wall thickness and left ventricular anterior wall dimensions at both diastole and systole.[182] ^73 TMAO can induce the expression of inflammatory factors and has obvious proinflammatory effects. The inflammatory response associated with the development of hypertension is an important factor in the occurrence of target organ damage, such as LVH. Furthermore, a decreased level of LA in patients with LVH was observed in our study. LA and α‐LA have a protective effect against high BP and helps reduce the risk of cardiovascular disease. A meta‐analysis showed that dietary LA intake is inversely associated with coronary heart disease risk in a dose–response manner.[183] ^74 We acknowledge that the present study has several limitations. Our sample size is relatively small. In the future, further studies with a larger sample size are warranted to truly understand the association between LVH and gut microbiota and metabolites. The present study also lacks mechanistic studies in animal models to determine the causality and role of gut microbiota on the development of LVH. Furthermore, information about exercise and diet, which may also have an impact on the gut microbiota, was not collected and corrected for in our study. Despite the limitations, our study identified an association between gut microbiota and its metabolites and LVH in clinical trials. Lack of early intervention leads to irreversible myocardial hypertrophy and interstitial fibrosis, resulting in impaired cardiac function and worsening long‐term outcomes. Our exploration is of great significance to provide new therapeutic ideas for other therapeutic options besides drug therapy in clinics, such as intestinal flora transplantation and metabolite supplementation. Our study can provide ideas for early intervention targets to prevent patients with hypertension from developing LVH and to provide means of reversal for patients who have already developed LVH. Sources of Funding This work was supported by the Clinical Research Special Fund of Wu Jieping Medical Foundation (320.6750.19089‐90). Disclosures None. Supporting information Tables S1–S10 [184]JAH3-13-e034230-s001.pdf^ (2.5MB, pdf) Figures S1–S15 [185]JAH3-13-e034230-s002.xlsx^ (46.5MB, xlsx) Acknowledgments